Synthesis and antimicrobial activity of novel 2,4-disubstituted thiazoles

Green chemistry

Proceedings of the 2nd International Scientific Conference «Chemical Technology and Engineering»: June 24–28, 2019, Lviv: Lviv Polytechnic National University, 2018, pp. 249–250

DOI: https://doi.org/10.23939/cte2019.01.249

Authors

First and Last Name	Academic degree	E-mail	Affiliation
Birutė Grybaitė	Ph.D.	birute.grybaite [at] ktu.edu	Kaunas University of Technology Kaunas, Lithuania
Rita Vaickelionienė	Ph.D.	vymic [at] ktu.lt	Kaunas University of Technology Kaunas, Lithuania
Vytautas Mickevičius	Sc.D.	vytautas.mickevicius [at] ktu.lt	Kaunas University of Technology Kaunas , Lithuania
Volodymyr Novikov	Sc.D.	volodymyr.p.novikov [at] lpnu.ua	Lviv Polytechnic National University Lviv , Ukraine
Viktor Zvarych	Ph.D.	maryna.v.stasevych [at] lpnu.ua	Lviv Polytechnic National University Lviv, Ukraine

I and my co-authors (if any) authorize the use of the Paper in accordance with the Creative Commons CC BY license

First published on this website: 15.03.2019 - 14:03

Abstract

A beneficial modifications of 2-substituted thiazoles by incorporating different functional groups into the structure such as carboxyl, chloromethyl, (phenylamino)methyl, ethoxyoxoethyl, which determine a certain chemical reactions of the compound was developed. All the synthesized compounds were tested for their in vitro antimicrobial and antifungal activity.

Keywords

amino acids antimicrobial agents cyclization functionalized thiazoles reactive intermediates

References

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